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Cat. No. Product Name Target Signaling Pathways
TP1260 [Pyr1]-Apelin-13

[pGlu1]-Apelin-13,人牛吡啶APELIN-13

Apelin receptor GPCR/G Protein
[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) 是一种高效的、内源性 apelin 受体选择性激动剂。
TP2001 MM 54

Potent apelin receptor antagonist (Ki = 82 nM; IC50 = 93 nM). Antagonizes the inhibitory affect of [Pyr1]-Apelin-13 on forskolin-induced cAMP accumulation in CHO-K1-APJ cells. Recuces tumor expansion and lengthens survival time in a mouse xenograft model

化合物

[Pyr1]-Apelin-13
Cat.No: TP1260
Synonym: [pGlu1]-Apelin-13,人牛吡啶APELIN-13
Target: Apelin receptor
MM 54
Cat.No: TP2001
Synonym:
Target:
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